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Le, Thuy, Kundu, Abhijit, Ghoshal, Atanu, Nguyen, Nghi, Preston, Sarah, Jiao, Yaqing, Ruan, Banfeng, Xue, Lian, Huang, Fei, Keiser, Jennifer, Hofmann, Andreas, Chang, Bill, Garcia-Bustos, Jose, Wells, Timothy, Palmer, Michael, Jabbar, Abdul, Gasser, Robin, Baell, Jonathan. ACS Publications; 2019. Structure-activity relationship studies of tolfenpyrad reveal subnanomolar inhibitors of haemonchus contortus development.
Hofmann, Andreas, Preston, Sarah, Cross, Megan, Herath, Dilrukshi, Simon, Anne, Gasser, Robin. BMC; 2019. DRfit : A Java tool for the analysis of discrete data from multi-well plate assays.
Jiao, Yaqing, Preston, Sarah, Song, Hongjian, Jabbar, Abdul, Liu, Yuxiu, Baell, Jonathan, Hofmann, Andreas, Hutchinson, Dana, Wang, Tao, Koehler, Anson, Fisher, Gillian, Andrews, Katherine, Laleu, Benoit, Palmer, Michael, Burrows, Jeremy, Wells, Timothy, Wang, Qingmin, Gasser, Robin. BioMed Central Ltd.; 2017. Assessing the anthelmintic activity of pyrazole-5-carboxamide derivatives against Haemonchus contortus.
Herath, Dilrukshi, Song, Hongjian, Preston, Sarah, Jabbar, Abdul, Wang, Tao, McGee, Sean, Hofmann, Andreas, Garcia-Bustos, Jose, Chang, Bill, Koehler, Anson, Liu, Yuxiu, Ma, Qiaoqiao, Zhang, Penqxiang, Zhao, Qiqi, Wang, Qingmin, Gasser, Robin. Elsevier Ltd; 2018. Arylpyrrole and fipronil analogues that inhibit the motility and/or development of Haemonchus contortus in vitro.
Kumarasingha, Rasika, Karpe, Avinash, Preston, Sarah, Yeo, Tiong-Chia, Lim, Diana, Tu, Chu-Lee, Luu, Jennii, Simpson, Kaylene, Shaw, Jillian, Gasser, Robin, Beale, David, Morrison, Paul, Palombo, Enzo, Boag, Peter. ; 2016. Metabolic profiling and in vitro assessment of anthelmintic fractions of Picria fel-terrae Lour.
Nguyen, Linh, Kurz, Thomas, Preston, Sarah, Brueckmann, Hjoerdis, Lungerich, Beate, Herath, Dilrukshi, Koehler, Anson, Wang, Tao, Skalova, Lenka, Jabbar, Abdul, Gasser, Robin. BMC; 2019. Phenotypic screening of the 'Kurz-box' of chemicals identifies two compounds (BLK127 and HBK4) with anthelmintic activity in vitro against parasitic larval stages of Haemonchus contortus.
Preston, Sarah, Luo, Junjie, Zhang, Yuezhou, Jabbar, Abdul, Crawford, Simon, Baell, Jonathan, Hofmann, Andreas, Hu, Min, Zhou, Hai-Bing, Gasser, Robin. BMC; 2016. Selenophene and thiophene-core estrogen receptor ligands that inhibit motility and development of parasitic stages of Haemonchus contortus.
Preston, Sarah, Jiao, Yaqing, Baell, Jonathan, Keiser, Jennifer, Crawford, Simon, Koehler, Anson, Wang, Tao, Simpson, Moana, Kaplan, Ray, Cowley, Karla, Simpson, Kaylene, Hofmann, Andreas, Jabbar, Abdul, Gasser, Robin. Elsevier Ltd; 2017. Screening of the ‘Open Scaffolds’ collection from Compounds Australia identifies a new chemical entity with anthelmintic activities against different developmental stages of the barber's pole worm and other parasitic nematodes.
Preston, Sarah, Korhonen, Pasi, Mouchiroud, Laurent, Cornaglia, Matteo, McGee, Sean, Young, Neil, Davis, Rohan, Crawford, Simon, Nowell, Cameron, Ansell, Brendan, Fisher, Gillian, Andrews, Katherine, Chang, Bill, Gijs, Martin, Sternberg, Paul, Auwerx, Johan, Baell, Jonathan, Hofmann, Andreas, Jabbar, Abdul, Gasser, Robin. FASEB; 2017. Deguelin exerts potent nematocidal activity via the mitochondrial respiratory chain.
Herath, Dilrukshi, Preston, Sarah, Hofmann, Andreas, Davis, Rohan, Koehler, Anson, Chang, Bill, Jabbar, Abdul, Gasser, Robin. Elsevier B.V.; 2017. Screening of a small, well-curated natural product-based library identifies two rotenoids with potent nematocidal activity against Haemonchus contortus.
Preston, Sarah, Jabbar, Abdul, Nowell, Cameron, Joachim, Anja, Ruttkowski, Barbel, Baell, Jonathan, Cardno, Tony, Korhonen, Pasi, Piedrafita, David, Ansell, Brendan, Jex, Aaron, Hofmann, Andreas, Gasser, Robin. Elsevier Ltd; 2015. Low cost whole-organism screening of compounds for anthelmintic activity.
Preston, Sarah, Jabbar, Abdul, Gasser, Robin. Elsevier B.V.; 2016. A perspective on genomic-guided anthelmintic discovery and repurposing using Haemonchus contortus.
Herath, Dilrukshi, Preston, Sarah, Jabbar, Abdul, Garcia-Bustos, Jose, Addison, Russell, Hayes, Sasha, Rali, Topul, Wang, Tao, Koehler, Anson, Chang, Bill, Hofmann, Andreas, Davis, Rohan, Gasser, Robin. Elsevier; 2019. Selected alpha-pyrones from the plants Cryptocarya novoguineensis (Lauraceae) and Piper methysticum (Piperaceae) with activity against Haemonchus contortus in vitro.
Sakthivel, Dhanasekaran, Swan, Jaclyn, Preston, Sarah, Shakif-Azam, MD, Faou, Pierre, Jiao, Yaqing, Downs, Rachael, Rajapaksha, Harinda, Gasser, Robin, Piedrafita, David, Beddoe, Travis. Peerj Inc.; 2018. Proteomic identification of galectin-11 and 14 ligands from Haemonchus contortus.
Le, Thuy, Kundu, Abhijit, Ghoshal, Atanu, Nguyen, Nghi, Preston, Sarah, Jiao, Yaqing, Ruan, Banfeng, Xue, Lian, Huang, Fei, Keiser, Jennifer, Hofmann, Andreas, Chang, Bill, Garcia-Bustos, Jose, Wells, Timothy, Palmer, Michael, Jabbar, Abdul, Gasser, Robin, Baell, Jonathan. ACS Publications; 2019. Novel 1-Methyl-1H-pyrazole-5-carboxamide derivatives with potent anthelmintic activity.
Jiao, Yaqing, Preston, Sarah, Hofmann, Andreas, Taki, Aya, Baell, Jonathan, Chang, Bill, Jabbar, Abdul, Gasser, Robin. Academic Press; 2020. A perspective on the discovery of selected compounds with anthelmintic activity against the barber's pole worm—Where to from here?.
Kumarasingha, Rasika, Preston, Sarah, Yeo, Tiong-Chia, Lim, Diana, Tu, Chu-Lee, Palombo, Enzo, Shaw, Jillian, Gasser, Robin, Boag, Peter. BioMed Central Ltd.; 2016. Anthelmintic activity of selected ethno-medicinal plant extracts on parasitic stages of Haemonchus contortus.
Herath, Dilrukshi, Preston, Sarah, Jabbar, Abdul, Garcia-Bustos, Jose, Taki, Aya, Addison, Russell, Hayes, Sasha, Beattie, Karren, McGee, Sean, Martin, Sheree, Ekin, Merrick, Hooper, John, Chang, Bill, Hofmann, Andreas, Davis, Rohan, Gasser, Robin. MDPI AG; 2019. Identification of fromiamycalin and halaminol A from Australian marine sponge extracts with anthelmintic activity against haemonchus contortus.
Le, Thuy, Kunda, Abhijit, Ghoshal, Atanu, Preston, Sarah, Jiao, Yaqing, Ruan, Banfeng, Xue, Lian, Huang, Fei, Keiser, Jennifer, Hofmann, Andreas, Chang, Bill, Garcia-Bustos, Jose, Jabbar, Abdul, Wells, Timothy, Palmer, Michael, Gasser, Robin, Baell, Jonathan. American Chemical Society; 2018. Optimization of novel 1-Methyl-1H-Pyrazole-5-carboxamides leads to high potency larval development inhibitors of the Barber's pole worm.
Ruan, Banfeng, Zhang, Yuezhou, Tadesse, Solomon, Preston, Sarah, Taki, Aya, Jabbar, Abdul, Hofmann, Andreas, Jiao, Yaqing, Garcia-Bustos, Jose, Harjani, Jitendra, Le, Thuy, Varghese, Swapna, Teguh, Silvia, Xie, Yiyue, Odiba, Jephthah, Hu, Min, Gasser, Robin, Baell, Jonathan. Elsevier Masson SAS; 2020. Synthesis and structure-activity relationship study of pyrrolidine-oxadiazoles as anthelmintics against Haemonchus contortus.
Herath, H. M. P. Dilrukshi, Taki, Aya, Sleebs, Brad, Hofmann, Andreas, Nguyen, Nghi, Preston, Sarah, Davis, Rohan, Jabbar, Abdul, Gasser, Robin. Academic Press; 2021. Advances in the discovery and development of anthelmintics by harnessing natural product scaffolds.
Sakthivel, Dhanasekaran, Preston, Sarah, Gasser, Robin, Meeusen, Els, Piedrafita, David. Nature Research; 2020. The oligomeric assembly of galectin-11 is critical for anti-parasitic activity in sheep (Ovis aries).
Li, Facai, Lok, James, Gasser, Robin, Korhonen, Pasi, Sandeman, Mark, Shi, Deshi, Zhou, Rui, Li, Xiangrui, Zhou, Yanqin, Zhao, Junlong, Hu, Min. Elsevier Ltd; 2014. Hc-daf-2 encodes an insulin-like receptor kinase in the barber's pole worm, Haemonchus contortus, and restores partial dauer regulation.